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Showing results 1 to 20 of 34
DateTitleAuthor(s)Full text
2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
2011Synthesis of variously coupled conjugates of D-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylaseKun, Sandor; Nagy, Gergo Z.; Toth, Marietta; Czecze, Laura; Albert Nguyen Van Nhien; Docsa, Tibor; Gergely, Pal; Charavgi, Maria-Despoina; Skourti, Paraskevi V.; Chrysina, Evangelia D.; Patonay, Tamas; Somsak, Laszlo
2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
2011From Structure-Based to Knowledge-Based Drug Design Through X-Ray Protein Crystallography: Sketching Glycogen Phosphorylase Binding SitesChrysina, E. D.; Chajistamatiou, A.; Chegkazi, M.
2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
2010The Prototype of Glycogen PhosphorylaseChrysina, E. D.
2010Glycogen phosphorylase inhibitor identification targeting the inhibitor binding site using virtual screening and experimental validationZhong, Shijun; Alexacou, Kyra-Melinda; Charavgi, Marianna A.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; MacKerell, Alexander D., Jr.
2010Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitorsFelfoldi, Nora; Toth, Marietta; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Alexacou, Kyra-Melinda; Somsak, Laszlo
2009Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitorsBenltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Chrysina, Evangelia D.; Zographos, Spyros E.; Leonidas, Demetres D.; Archontis, Georgios; Oikonomakos, Nikos G.
2009Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase caseChrysina, Evangelia D.; Bokor, Eva; Alexacou, Kyra-Melinda; Charavgi, Maria-Despoina; Oikonomakos, George N.; Zographos, Spyros E.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Laszlo, Somsak
2008New Inhibitors of Glycogen Phosphorylase as Potential Antidiabetic AgentsSomsak, L.; Czifrak, K.; Toth, M.; Bokor, E.; Chrysina, E. D.; Alexacou, K. -M.; Hayes, J. M.; Tiraidis, C.; Lazoura, E.; Leonidas, D. D.; Zographos, S. E.; Oikonomakos, N. G.
2008Crystallographic and computational studies on 4-phenyl-N-(beta-D-glucopyranosyl)-1H-1,2, 3-triazole-1-acetamide, an inhibitor of glycogen phosphorylase: Comparison with alpha-D-glucose, N-acetyl-beta-D-glucopyranosylamine and N-benzoyl-N '-beta-D-glucopyranosyl urea bindingAlexacou, Kyra-Melinda; Hayes, Joseph M.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Archontis, Georgios; Oikonomakos, Nikos G.; Paul, Jashuva V.; Varghese, Babu; Loganathan, Duraikkannu
2007In the search of glycogen phosphorylase inhibitors: 4. Synthesis of C-D-glycopyranosylbenzo(hydro)quinones - Inhibition of and binding to glycogen phosphorylase in the crystalHe, L.; Zhang, Y. Z.; Tanoh, M.; Chen, G. R.; Praly, J. P.; Chrysina, Evangelia D.; Tiraidis, C.; Kosmopoulou, M.; Leonidas, Demetres D.; Oikonomakos, Nikos G.
2006Indirubin and indigo analogues as potential inhibitors of glycogenolysis: structural basis of glycogen phosphorylase inhibitionOikonomakos, Nikos G.; Kosmopoulou, Magda N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Tiraidis, Costas; Bischler, Nicolas; Tsitsanou, Katerina E.; Zographos, Spyros E.; Kostas, Ioannis D.; Eisenbrand, Gerhard
2006Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-D-glucopyranosylamine and N-trifluoroacetyl-beta-D-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylaseAnagnostou, E.; Kosmopoulou, M. N.; Chrysina, Evangelia D.; Leonidas, D. D.; Hadjiloi, T.; Tiraidis, C.; Zographos, S. E.; Gyorgydeak, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Kolisis, Fragiskos N.; Oikonomakos, Nikos G.
2006Crystallographic studies on N-azidoacetyl-beta-D-glucopyranosylamine, an inhibitor of glycogen phosphorylase: Comparison with N-acetyl-beta-D-glucopyranosylaminePetsalakis, E. I.; Chrysina, Evangelia D.; Tiraidis, C.; Hadjiloi, T.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Aich, U.; Varghese, B.; Loganathan, D.
2006Binding of oxalyl derivatives of beta-D-glucopyranosylamine to muscle glycogen phosphorylase bHadjiloi, T.; Tiraidis, C.; Chrysina, Evangelia D.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Tsipos, P.; Gimisis, T.
2005Indirubin-3 '-aminooxy-acetate inhibits glycogen phosphorylase by binding at the inhibitor and the allosteric site. Broad specificities of the two sitesKosmopoulou, M. N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Eisenbrand, G.; Oikonomakos, Nikos G.
2005Kinetic and crystallographic studies of glucopyranose spirohydantoin and glucopyranosylamine analogs inhibitors of glycogen phosphorylaseWatson, K. A.; Chrysina, Evangelia D.; Tsitsanou, K. E.; Zographos, Spyros E.; Archontis, G.; Fleet, G. W. J.; Oikonomakos, Nikos G.
2005Kinetic and crystallographic studies on 2-(beta-D-glucopyranosyl)-5-methyl-1,3,4-oxadiazole, -benzothiazole, and -benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding siteChrysina, Evangelia D.; Kosmopoulou, M. N.; Tiraidis, C.; Kardakaris, R.; Bischler, N.; Leonidas, Demetres D.; Hadady, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Oikonomakos, Nikos G.
Showing results 1 to 20 of 34

 

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