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Showing results 1 to 20 of 34
| Date | Title | Author(s) | Full text | | 2012 | N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods | Veronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak | |
| 2011 | Synthesis of variously coupled conjugates of D-glucose, 1,3,4-oxadiazole, and 1,2,3-triazole for inhibition of glycogen phosphorylase | Kun, Sandor; Nagy, Gergo Z.; Toth, Marietta; Czecze, Laura; Albert Nguyen Van Nhien; Docsa, Tibor; Gergely, Pal; Charavgi, Maria-Despoina; Skourti, Paraskevi V.; Chrysina, Evangelia D.; Patonay, Tamas; Somsak, Laszlo | |
| 2011 | Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylase | Alexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D. | |
| 2011 | From Structure-Based to Knowledge-Based Drug Design Through X-Ray Protein Crystallography: Sketching Glycogen Phosphorylase Binding Sites | Chrysina, E. D.; Chajistamatiou, A.; Chegkazi, M. | |
| 2010 | The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitors | Alexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D. | |
| 2010 | The Prototype of Glycogen Phosphorylase | Chrysina, E. D. | |
| 2010 | Glycogen phosphorylase inhibitor identification targeting the inhibitor binding site using virtual screening and experimental validation | Zhong, Shijun; Alexacou, Kyra-Melinda; Charavgi, Marianna A.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; MacKerell, Alexander D., Jr. | |
| 2010 | Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitors | Felfoldi, Nora; Toth, Marietta; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Alexacou, Kyra-Melinda; Somsak, Laszlo | |
| 2009 | Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitors | Benltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Chrysina, Evangelia D.; Zographos, Spyros E.; Leonidas, Demetres D.; Archontis, Georgios; Oikonomakos, Nikos G. | |
| 2009 | Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase case | Chrysina, Evangelia D.; Bokor, Eva; Alexacou, Kyra-Melinda; Charavgi, Maria-Despoina; Oikonomakos, George N.; Zographos, Spyros E.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Laszlo, Somsak | |
| 2008 | New Inhibitors of Glycogen Phosphorylase as Potential Antidiabetic Agents | Somsak, L.; Czifrak, K.; Toth, M.; Bokor, E.; Chrysina, E. D.; Alexacou, K. -M.; Hayes, J. M.; Tiraidis, C.; Lazoura, E.; Leonidas, D. D.; Zographos, S. E.; Oikonomakos, N. G. | |
| 2008 | Crystallographic and computational studies on 4-phenyl-N-(beta-D-glucopyranosyl)-1H-1,2, 3-triazole-1-acetamide, an inhibitor of glycogen phosphorylase: Comparison with alpha-D-glucose, N-acetyl-beta-D-glucopyranosylamine and N-benzoyl-N '-beta-D-glucopyranosyl urea binding | Alexacou, Kyra-Melinda; Hayes, Joseph M.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Archontis, Georgios; Oikonomakos, Nikos G.; Paul, Jashuva V.; Varghese, Babu; Loganathan, Duraikkannu | |
| 2007 | In the search of glycogen phosphorylase inhibitors: 4. Synthesis of C-D-glycopyranosylbenzo(hydro)quinones - Inhibition of and binding to glycogen phosphorylase in the crystal | He, L.; Zhang, Y. Z.; Tanoh, M.; Chen, G. R.; Praly, J. P.; Chrysina, Evangelia D.; Tiraidis, C.; Kosmopoulou, M.; Leonidas, Demetres D.; Oikonomakos, Nikos G. | |
| 2006 | Crystallographic studies on N-azidoacetyl-beta-D-glucopyranosylamine, an inhibitor of glycogen phosphorylase: Comparison with N-acetyl-beta-D-glucopyranosylamine | Petsalakis, E. I.; Chrysina, Evangelia D.; Tiraidis, C.; Hadjiloi, T.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Aich, U.; Varghese, B.; Loganathan, D. | |
| 2006 | Binding of oxalyl derivatives of beta-D-glucopyranosylamine to muscle glycogen phosphorylase b | Hadjiloi, T.; Tiraidis, C.; Chrysina, Evangelia D.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Tsipos, P.; Gimisis, T. | |
| 2006 | Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-D-glucopyranosylamine and N-trifluoroacetyl-beta-D-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylase | Anagnostou, E.; Kosmopoulou, M. N.; Chrysina, Evangelia D.; Leonidas, D. D.; Hadjiloi, T.; Tiraidis, C.; Zographos, S. E.; Gyorgydeak, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Kolisis, Fragiskos N.; Oikonomakos, Nikos G. | |
| 2006 | Indirubin and indigo analogues as potential inhibitors of glycogenolysis: structural basis of glycogen phosphorylase inhibition | Oikonomakos, Nikos G.; Kosmopoulou, Magda N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Tiraidis, Costas; Bischler, Nicolas; Tsitsanou, Katerina E.; Zographos, Spyros E.; Kostas, Ioannis D.; Eisenbrand, Gerhard | |
| 2005 | Glycogen phosphorylase inhibitors: A free energy perturbation analysis of glucopyranose spirohydantoin analogues | Archontis, G.; Watson, K. A.; Xie, Q.; Andreou, G.; Chrysina, Evangelia D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Karplus, M. | |
| 2005 | Binding of beta-D-glucopyranosyl bismethoxyphosphoramidate to glycogen phosphorylase b: kinetic and crystallographic studies | Chrysina, Evangelia D.; Kosmopoulou, M. N.; Kardakaris, R.; Bischler, N.; Leonidas, Demetres D.; Kannan, T.; Loganathan, D.; Oikonomakos, Nikos G. | |
| 2005 | Kinetic and crystallographic studies on 2-(beta-D-glucopyranosyl)-5-methyl-1,3,4-oxadiazole, -benzothiazole, and -benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding site | Chrysina, Evangelia D.; Kosmopoulou, M. N.; Tiraidis, C.; Kardakaris, R.; Bischler, N.; Leonidas, Demetres D.; Hadady, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Oikonomakos, Nikos G. |  |
Showing results 1 to 20 of 34
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