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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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1996Glucofuranose analogues of hydantocidinBrandstetter, T. W.; delaFuente, C.; Kim, Y. H.; Johnson, L. N.; Crook, S.; Lilley, Pmdq; Watkin, D. J.; Tsitsanou, K. E.; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Fleet, G. W. J.
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1997The structure of glycogen phosphorylase b with an alkyl-dihydropyridine-dicarboxylic acid compound, a novel and potent inhibitorZographos, Spyros E.; Oikonomakos, Nikos G.; Tsitsanou, K. E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Skamnaki, V. T.; Bischoff, H.; Goldmann, S.; Watson, K. A.; Johnson, L. N.
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2002Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b - Kinetic and crystallographic studiesOikonomakos, Nikos G.; Kosmopoulou, M.; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Somsak, U.; Nagy, V.; Praly, J. P.; Docsa, T.; Toth, A.; Gergely, P.
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2003Crystal structure of rabbit muscle glycogen phosphorylase a in complex with a potential hypoglycaemic drug at 2.0 angstrom resolutionOikonomakos, Nikos G.; Chrysina, Evangelia D.; Kosmopoulou, M. N.; Leonidas, Demetres D.
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2003Crystallization and preliminary X-ray crystallographic analysis of Sclerotium rolfsii lectinLeonidas, Demetres D.; Swamy, B. M.; Bhat, A. G.; Inamdar, S. R.; Kosmopoulou, M. N.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.
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2003High-resolution crystal structures of ribonuclease A complexed with adenylic and uridylic nucleotide inhibitors. Implications for structure-based design of ribonucleolytic inhibitorsLeonidas, Demetres D.; Chavali, G. B.; Oikonomakos, Nikos G.; Chrysina, Evangelia D.; Kosmopoulou, M. N.; Vlassi, M.; Frankling, C.; Acharya, K. R.
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2003Crystallographic studies on alpha- and beta-D-glucopyranosyl formamide analogues, inhibitors of glycogen phosphorylaseChrysina, Evangelia D.; Oikonomakos, Nikos G.; Zographos, Spyros E.; Kosmopoulou, M. N.; Bischler, N.; Leonidas, Demetres D.; Kovacs, L.; Docsa, T.; Gergely, P.; Somsak, L.
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2003The binding of beta- and gamma-cyclodextrins to glycogen phosphorylase b: Kinetic and crystallographic studiesPinotsis, N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Mavridis, I. M.
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2004Ορθολογιστικός σχεδιασμός νέων υπογλυκαιμικών φαρμάκωνLeonidas, Demetres D.; Chrysina, Evangelia D.; Κοσμοπούλου, Μάγδα Ν.; Καρδακάρη, Ροζίνα; Oikonomakos, Nikos G.; Bischler, Nicolas
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2004Binding of the potential antitumour agent indirubin-5-sulphonate at the inhibitor site of rabbit muscle glycogen phosphorylase b - Comparison with ligand binding to pCDK2-cyclin A complexKosmopoulou, M. N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Bischler, N.; Eisenbrand, G.; Sakarellos, C. E.; Pauptit, R.; Oikonomakos, Nikos G.
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2004Kinetic and modelling studies on the lipase catalysed enantio selective esterification of (+/-)-perillyl alcoholSkouridou, V.; Chrysina, Evangelia D.; Stamatis, H.; Oikonomakos, Nikos G.; Kolisis, Fragiskos N.‏
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2005Glycogen phosphorylase inhibitors: A free energy perturbation analysis of glucopyranose spirohydantoin analoguesArchontis, G.; Watson, K. A.; Xie, Q.; Andreou, G.; Chrysina, Evangelia D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Karplus, M.
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2005Indirubin-3 '-aminooxy-acetate inhibits glycogen phosphorylase by binding at the inhibitor and the allosteric site. Broad specificities of the two sitesKosmopoulou, M. N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Eisenbrand, G.; Oikonomakos, Nikos G.
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2005Kinetic and crystallographic studies on 2-(beta-D-glucopyranosyl)-5-methyl-1,3,4-oxadiazole, -benzothiazole, and -benzimidazole, inhibitors of muscle glycogen phosphorylase b. Evidence for a new binding siteChrysina, Evangelia D.; Kosmopoulou, M. N.; Tiraidis, C.; Kardakaris, R.; Bischler, N.; Leonidas, Demetres D.; Hadady, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Oikonomakos, Nikos G.
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2005Kinetic and crystallographic studies of glucopyranose spirohydantoin and glucopyranosylamine analogs inhibitors of glycogen phosphorylaseWatson, K. A.; Chrysina, Evangelia D.; Tsitsanou, K. E.; Zographos, Spyros E.; Archontis, G.; Fleet, G. W. J.; Oikonomakos, Nikos G.
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2005Binding of beta-D-glucopyranosyl bismethoxyphosphoramidate to glycogen phosphorylase b: kinetic and crystallographic studiesChrysina, Evangelia D.; Kosmopoulou, M. N.; Kardakaris, R.; Bischler, N.; Leonidas, Demetres D.; Kannan, T.; Loganathan, D.; Oikonomakos, Nikos G.
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2005Crystallographic studies on acyl ureas, a new class of glycogen phosphorylase inhibitors, as potential antidiabetic drugsOikonomakos, Nikos G.; Kosmopoulou, M. N.; Chrysina, Evangelia D.; Leonidas, Demetres D.; Kostas, Ioannis D.; Wendt, K. U.; Klabunde, T.; Defossa, E.
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2006Crystallographic studies on N-azidoacetyl-beta-D-glucopyranosylamine, an inhibitor of glycogen phosphorylase: Comparison with N-acetyl-beta-D-glucopyranosylaminePetsalakis, E. I.; Chrysina, Evangelia D.; Tiraidis, C.; Hadjiloi, T.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Aich, U.; Varghese, B.; Loganathan, D.
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2006Binding of oxalyl derivatives of beta-D-glucopyranosylamine to muscle glycogen phosphorylase bHadjiloi, T.; Tiraidis, C.; Chrysina, Evangelia D.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Tsipos, P.; Gimisis, T.
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2006Crystallographic studies on two bioisosteric analogues, N-acetyl-beta-D-glucopyranosylamine and N-trifluoroacetyl-beta-D-glucopyranosylamine, potent inhibitors of muscle glycogen phosphorylaseAnagnostou, E.; Kosmopoulou, M. N.; Chrysina, Evangelia D.; Leonidas, Demetres D.; Hadjiloi, T.; Tiraidis, C.; Zographos, Spyros E.; Gyorgydeak, Z.; Somsak, L.; Docsa, T.; Gergely, P.; Kolisis, Fragiskos N.‏; Oikonomakos, Nikos G.
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