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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2009Morpholino, Piperidino, and Pyrrolidino Derivatives of Pyrimidine Nucleosides as Inhibitors of Ribonuclease A: Synthesis, Biochemical, and Crystallographic EvaluationSamanta, Anirban; Leonidas, Demetres D.; Dasgupta, Swagata; Pathak, Tanmaya; Zographos, Spyros E.; Oikonomakos, Nikos G.
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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20101-(3-Deoxy-3-fluoro-beta-D-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studiesTsirkone, Vicky G.; Tsoukala, Evangelia; Lamprakis, Christos; Manta, Stella; Hayes, Joseph M.; Skamnaki, Vicky T.; Drakou, Christina; Zographos, Spyros E.; Komiotis, Dimitri; Leonidas, Demetres D.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2002Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b - Kinetic and crystallographic studiesOikonomakos, Nikos G.; Kosmopoulou, M.; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Somsak, U.; Nagy, V.; Praly, J. P.; Docsa, T.; Toth, A.; Gergely, P.
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1994The design of potential antidiabetic drugs: Experimental investigation of a number of ?-D-glucose analogue inhibitors of glycogen phosphorylaseOikonomakos, Nikos G.; Kontou, M.; Zographos, Spyros E.; Tsitoura, H. S.; Johnson, L. N.; Watson, K. A.; Mitchell, E. P.; Fleet, G. W. J.; Son, J. C.; Bichard, C. J. F.; Leonidas, Demetres D.; Acharya, K. R.
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2007FR258900, a potential anti-hyperglycemic drug, binds at the allosteric site of glycogen phosphorylaseTiraidis, C.; Alexacou, K. M.; Zographos, Spyros E.; Leonidas, Demetres D.; Gimisis, T.; Oikonomakos, Nikos G.
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1994The Design of Potential Antidiabetic Drugs - Experimental Investigation of a Number of Beta-D-Glucose Analog Inhibitors of Glycogen-PhosphorylaseOikonomakos, Nikos G.; Kontou, M.; Zographos, Spyros E.; Tsitoura, H. S.; Johnson, L. N.; Watson, K. A.; Mitchell, E. P.; Fleet, G. W. J.; Son, J. C.; Bichard, C. J. F.; Leonidas, Demetres D.; Acharya, K. R.
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1997The structure of glycogen phosphorylase b with an alkyl-dihydropyridine-dicarboxylic acid compound, a novel and potent inhibitorZographos, Spyros E.; Oikonomakos, Nikos G.; Tsitsanou, K. E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Skamnaki, V. T.; Bischoff, H.; Goldmann, S.; Watson, K. A.; Johnson, L. N.
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1995Sulfate-Activated Phosphorylase-B - the Ph-Dependence of Catalytic ActivityZographos, Spyros E.; Oikonomakos, Nikos G.; Dixon, H. B. F.; Griffin, W. G.; Johnson, L. N.; Leonidas, Demetres D.
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