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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2002Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b - Kinetic and crystallographic studiesOikonomakos, Nikos G.; Kosmopoulou, M.; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Somsak, U.; Nagy, V.; Praly, J. P.; Docsa, T.; Toth, A.; Gergely, P.
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1999Allosteric inhibition of glycogen phosphorylase a by the potential antidiabetic drug 3-isopropyl 4-(2-chlorophenyl)-1,4-dihydro-1-ethyl-2-methyl-pyridine-3,5,6-tricarbox ylateOikonomakos, Nikos G.; Tsitsanou, K. E.; Zographos, Spyros E.; Skamnaki, V. T.; Goldmann, S.; Bischoff, H.
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1999Molecular recognition in glycogen phosphorylase inhibitor designTsitsanou, K. E.; Zographos, Spyros E.; Skamnaki, V. T.; Oikonomakos, Nikos G.
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1996A galactopyranose analogue of hydantocidinBrandstetter, T. W.; Wormald, M. R.; Dwek, R. A.; Butters, T. D.; Platt, F. M.; Tsitsanou, K. E.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Fleet, G. W. J.
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1995The Binding of 2-Deoxy-D-Glucose 6-Phosphate to Glycogen-Phosphorylase-B - Kinetic and Crystallographic StudiesOikonomakos, Nikos G.; Zographos, Spyros E.; Johnson, L. N.; Papageorgiou, A. C.; Acharya, K. R.
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1995Glucose Analog Inhibitors of Glycogen-Phosphorylase - from Crystallographic Analysis to Drug Prediction Using Grid Force-Field and Golpe Variable SelectionWatson, K. A.; Mitchell, E. P.; Johnson, L. N.; Cruciani, G.; Son, J. C.; Bichard, C. J. F.; Fleet, G. W. J.; Oikonomakos, Nikos G.; Kontou, M.; Zographos, Spyros E.
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1995Potent Inhibition of Glycogen-Phosphorylase by a Spirohydantoin of Glucopyranose - First Pyranose Analogs of HydantocidinBichard, C. J. F.; Mitchell, E. P.; Wormald, M. R.; Watson, K. A.; Johnson, L. N.; Zographos, Spyros E.; Koutra, D. D.; Oikonomakos, Nikos G.; Fleet, G. W. J.
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1997Triazole carboxylic acids as anionic sugar mimics? Inhibition of glycogen phosphorylase by a D-glucotriazole carboxylateKrulle, T.; delaFuente, C.; Pickering, L.; Aplin, R. T.; Tsitsanou, K. E.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Nash, R. J.; Griffiths, R. C.; Fleet, G. W. J.
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2000Flavopiridol inhibits glycogen phosphorylase by binding at the inhibitor siteOikonomakos, Nikos G.; Schnier, J. B.; Zographos, Spyros E.; Skamnaki, V. T.; Tsitsanou, K. E.; Johnson, L. N.
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2006Iminosugars as potential inhibitors of glycogenolysis: Structural insights into the molecular basis of glycogen phosphorylase inhibitionOikonomakos, Nikos G.; Tiraidis, C.; Leonidas, Demetres D.; Zographos, Spyros E.; Kristiansen, M.; Jessen, C. U.; Norskov-Lauritsen, L.; Agius, L.
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