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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2002Binding of N-acetyl-N '-beta-D-glucopyranosyl urea and N-benzoyl-N '-beta-D-glucopyranosyl urea to glycogen phosphorylase b - Kinetic and crystallographic studiesOikonomakos, Nikos G.; Kosmopoulou, M.; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Somsak, U.; Nagy, V.; Praly, J. P.; Docsa, T.; Toth, A.; Gergely, P.
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1994The design of potential antidiabetic drugs: Experimental investigation of a number of ?-D-glucose analogue inhibitors of glycogen phosphorylaseOikonomakos, Nikos G.; Kontou, M.; Zographos, Spyros E.; Tsitoura, H. S.; Johnson, L. N.; Watson, K. A.; Mitchell, E. P.; Fleet, G. W. J.; Son, J. C.; Bichard, C. J. F.; Leonidas, Demetres D.; Acharya, K. R.
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2007FR258900, a potential anti-hyperglycemic drug, binds at the allosteric site of glycogen phosphorylaseTiraidis, C.; Alexacou, K. M.; Zographos, Spyros E.; Leonidas, Demetres D.; Gimisis, T.; Oikonomakos, Nikos G.
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1994The Design of Potential Antidiabetic Drugs - Experimental Investigation of a Number of Beta-D-Glucose Analog Inhibitors of Glycogen-PhosphorylaseOikonomakos, Nikos G.; Kontou, M.; Zographos, Spyros E.; Tsitoura, H. S.; Johnson, L. N.; Watson, K. A.; Mitchell, E. P.; Fleet, G. W. J.; Son, J. C.; Bichard, C. J. F.; Leonidas, Demetres D.; Acharya, K. R.
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1997The structure of glycogen phosphorylase b with an alkyl-dihydropyridine-dicarboxylic acid compound, a novel and potent inhibitorZographos, Spyros E.; Oikonomakos, Nikos G.; Tsitsanou, K. E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Skamnaki, V. T.; Bischoff, H.; Goldmann, S.; Watson, K. A.; Johnson, L. N.
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1995Sulfate-Activated Phosphorylase-B - the Ph-Dependence of Catalytic ActivityZographos, Spyros E.; Oikonomakos, Nikos G.; Dixon, H. B. F.; Griffin, W. G.; Johnson, L. N.; Leonidas, Demetres D.
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2014Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: Synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methodsCzifrák K.; Páhi A.; Deák S.; Kiss-Szikszai A.; Kövér K.E.; Docsa T.; Gergely P.; Alexacou K.-M.; Papakonstantinou M.; Leonidas D.D.; Zographos S.E.; Chrysina E.D.; Somsák L.
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2013Structural analysis of the Rhizoctonia solani agglutinin reveals a domain-swapping dimeric assemblySkamnaki V.T.; Peumans W.J.; Kantsadi A.L.; Cubeta M.A.; Plas K.; Pakala S.; Zographos S.E.; Smagghe G.; Nierman W.C.; Van Damme E.J.M.; Leonidas D.D.
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2014Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-β-d-glucopyranosylaminesParmenopoulou V.; Kantsadi A.L.; Tsirkone V.G.; Chatzileontiadou D.S.M.; Manta S.; Zographos S.E.; Molfeta C.; Archontis G.; Agius L.; Hayes J.M.; Leonidas D.D.; Komiotis D.
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