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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2008New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferaseLi, Hongqing; Liu, Tao; Zhang, Yongmin; Favre, Sylvain; Bello, Claudia; Vogel, Pierre; Butters, Terry D.; Oikonomakos, Nikos G.; Marrot, Jerome; Bleriot, Yves
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2008Comparative docking studies of labdane-type diterpenes with forskolin at the active site of adenylyl cyclaseKoukoulitsa, Catherine; Zervou, Maria; Demetzos, Costas; Mavromoustakos, Thomas
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2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
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2012Synthesis of novel sulfonamide-1,2,4-triazoles, 1,3,4-thiadiazoles and 1,3,4-oxadiazoles, as potential antibacterial and antifungal agents. Biological evaluation and conformational analysis studiesZoumpoulakis, Panagiotis; Camoutsis, Ch.; Pairas, G.; Sokovic, M.; Glamoclija, J.; Potamitis, C.; Pitsas, A.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2011Regulation of the Escherichia coli AtoSC two component system by synthetic biologically active 5;7;8-trimethyl-1;4-benzoxazine analoguesFilippou, Panagiota S.; Koini, Eftychia N.; Calogeropoulou, Theodora; Kalliakmani, Panagiota; Panagiotidis, Christos A.; Kyriakidis, D.A.
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2010Novel 4-thiazolidinone derivatives as potential antifungal and antibacterial drugsOmar, Kouatli; Geronikaki, Athina; Zoumpoulakis, Panagiotis; Camoutsis, Charalabos; Sokovic, Marina; Ciric, Ana; Glamoclija, Jasmina
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2011Strategies in the Rational Drug DesignMavromoustakos, Thomas; Durdagi, S.; Koukoulitsa, C.; Simcic, M.; Papadopoulos, Manthos G.; Hodoscek, M.; Grdadolnik, S. Golic
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2011From Structure-Based to Knowledge-Based Drug Design Through X-Ray Protein Crystallography: Sketching Glycogen Phosphorylase Binding SitesChrysina, Evangelia D.; Chajistamatiou, A.; Chegkazi, M.
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