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| Τύπος | Ημερομηνία | Τίτλος | Δημιουργός | Πλήρες κείμενο |
| 2009 | Mapping the ribonucleolytic active site of bovine seminal ribonuclease. The binding of pyrimidinyl phosphonucleotide inhibitors | Dossi, Kyriaki; Tsirkone, Vicky G.; Hayes, Joseph M.; Matousek, Josef; Pouckova, Pavla; Soucek, Josef; Zadinova, Marie; Zographos, Spyros E.; Leonidas, Demetres D. | |
| 2010 | 1-(3-Deoxy-3-fluoro-beta-D-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies | Tsirkone, Vicky G.; Tsoukala, Evangelia; Lamprakis, Christos; Manta, Stella; Hayes, Joseph M.; Skamnaki, Vicky T.; Drakou, Christina; Zographos, Spyros E.; Komiotis, Dimitri; Leonidas, Demetres D. | |
| 2010 | Glycogen phosphorylase inhibitor identification targeting the inhibitor binding site using virtual screening and experimental validation | Zhong, Shijun; Alexacou, Kyra-Melinda; Charavgi, Marianna A.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; MacKerell, Alexander D., Jr. | |
| 2010 | The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitors | Alexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D. | |
| 2011 | Kinetics, in silico docking, molecular dynamics, and MM-GBSA binding studies on prototype indirubins, KT5720, and staurosporine as phosphorylase kinase ATP-binding site inhibitors: The role of water molecules examined | Hayes, Joseph M.; Skamnaki, Vicky T.; Archontis, Georgios; Lamprakis, Christos; Sarrou, Josephine; Bischler, Nicolas; Skaltsounis, Alexios-Leandros; Zographos, Spyros E.; Oikonomakos, Nikos G. | |
| 2011 | Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylase | Alexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D. | |
| 2012 | hCINAP is an atypical mammalian nuclear adenylate kinase with an ATPase motif: Structural and functional studies | Drakou, Christina E.; Malekkou, Anna; Hayes, Joseph M.; Lederer, Carsten W.; Leonidas, Demetres D.; Oikonomakos, Nikos G.; Lamond, Angus I.; Santama, Niovi; Zographos, Spyros E. | |
| 2012 | Anopheles gambiae odorant binding protein crystal complex with the synthetic repellent DEET: implications for structure-based design of novel mosquito repellents | Tsitsanou, K. E.; Thireou, T.; Drakou, C. E.; Koussis, K.; Keramioti, M. V.; Leonidas, Demetres D.; Eliopoulos, E.; Iatrou, K.; Zographos, Spyros E. | |
| 2012 | N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods | Veronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak | |
| 2012 | The s-Hole Phenomenon of Halogen Atoms Forms the Structural Basis of the Strong Inhibitory Potency of C5 Halogen Substituted Glucopyranosyl Nucleosides towards Glycogen Phosphorylase b | Kantsadi, Anastasia L.; Hayes, Joseph M.; Manta, Stella; Skamnaki, Vicky T.; Kiritsis, Christos; Psarra, Anna-Maria G.; Koutsogiannis, Zissis; Dimopoulou, Athina; Theofanous, Stavroula; Nikoleousakos, Nikolaos; Zoumpoulakis, Panagiotis; Kontou, Maria; Papadopoulos, George; Zographos, Spyros E.; Komiotis, Dimitris; Leonidas, Demetres D. | |
| 2012 | 3 '-Axial CH2OH Substitution on Glucopyranose does not Increase Glycogen Phosphorylase Inhibitory Potency. QM/MM-PBSA Calculations Suggest Why | Manta, Stella; Xipnitou, Andromachi; Kiritsis, Christos; Kantsadi, Anastassia L.; Hayes, Joseph M.; Skamnaki, Vicky T.; Lamprakis, Christos; Kontou, Maria; Zoumpoulakis, Panagiotis; Zographos, Spyros E.; Leonidas, Demetres D.; Komiotis, Dimitri | |
| 2013 | Structural analysis of the Rhizoctonia solani agglutinin reveals a domain-swapping dimeric assembly | Skamnaki V.T.; Peumans W.J.; Kantsadi A.L.; Cubeta M.A.; Plas K.; Pakala S.; Zographos S.E.; Smagghe G.; Nierman W.C.; Van Damme E.J.M.; Leonidas D.D. | |
| 2013 | Sourcing the affinity of flavonoids for the glycogen phosphorylase inhibitor site via crystallography, kinetics and QM/MM-PBSA binding studies: Comparison of chrysin and flavopiridol | Tsitsanou K.E.; Hayes J.M.; Keramioti M.; Mamais M.; Oikonomakos N.G.; Kato A.; Leonidas D.D.; Zographos S.E. | |
| 2013 | Crystal and solution studies of the "plus-C" odorant-binding protein 48 from Anopheles gambiae: Control of binding specificity through three-dimensional domain swapping | Tsitsanou K.E.; Drakou C.E.; Thireou T.; Gruber A.V.; Kythreoti G.; Azem A.; Fessas D.; Eliopoulos E.; Iatrou K.; Zographos S.E. | |
| 2014 | Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: Synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods | Czifrák K.; Páhi A.; Deák S.; Kiss-Szikszai A.; Kövér K.E.; Docsa T.; Gergely P.; Alexacou K.-M.; Papakonstantinou M.; Leonidas D.D.; Zographos S.E.; Chrysina E.D.; Somsák L. | |
| 2014 | Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-β-d-glucopyranosylamines | Parmenopoulou V.; Kantsadi A.L.; Tsirkone V.G.; Chatzileontiadou D.S.M.; Manta S.; Zographos S.E.; Molfeta C.; Archontis G.; Agius L.; Hayes J.M.; Leonidas D.D.; Komiotis D. | |
| 2015 | Molecular cloning, carbohydrate specificity and the crystal structure of two Sclerotium rolfsii lectin variants | Peppa V.I.; Venkat H.; Kantsadi A.L.; Inamdar S.R.; Bhat G.G.; Eligar S.; Shivanand A.; Chachadi V.B.; Satisha G.J.; Swamy B.M.; Skamnaki V.T.; Zographos S.E.; Leonidas D.D. | |
| 2016 | The crystal structure of the AgamOBP1•Icaridin complex reveals alternative binding modes and stereo-selective repellent recognition | Drakou C.E.; Tsitsanou K.E.; Potamitis C.; Fessas D.; Zervou M.; Zographos S.E. | |
| 2019 | Structural and biochemical studies of an odorant binding protein from the malaria vector anopheles gambiae | Liggri, P.; Tsitsanou, K.; Zographos, S. | |
| 2019 | Συνέντευξη τύπου: Pfizer και Εθνικό Ίδρυμα Ερευνών: Ισχυρή συμμαχία με στόχο την 'προαγωγή της επιστήμης' | Δήμας, Χρίστος; Gregoriou, Vasilis G.; Ραγκούσης, Ζαχαρίας; Pintzas, Alexander; Zographos, Spyros E. | |
