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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2008New Inhibitors of Glycogen Phosphorylase as Potential Antidiabetic AgentsSomsak, L.; Czifrak, K.; Toth, M.; Bokor, E.; Chrysina, Evangelia D.; Alexacou, K. -M.; Hayes, J. M.; Tiraidis, C.; Lazoura, E.; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.
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2009Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitorsBenltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Chrysina, Evangelia D.; Zographos, Spyros E.; Leonidas, Demetres D.; Archontis, Georgios; Oikonomakos, Nikos G.
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2010Synthesis of new glycosyl biuret and urea derivatives as potential glycoenzyme inhibitorsFelfoldi, Nora; Toth, Marietta; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Alexacou, Kyra-Melinda; Somsak, Laszlo
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20101-(3-Deoxy-3-fluoro-beta-D-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studiesTsirkone, Vicky G.; Tsoukala, Evangelia; Lamprakis, Christos; Manta, Stella; Hayes, Joseph M.; Skamnaki, Vicky T.; Drakou, Christina; Zographos, Spyros E.; Komiotis, Dimitri; Leonidas, Demetres D.
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2010The Prototype of Glycogen PhosphorylaseChrysina, Evangelia D.
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2011From Structure-Based to Knowledge-Based Drug Design Through X-Ray Protein Crystallography: Sketching Glycogen Phosphorylase Binding SitesChrysina, Evangelia D.; Chajistamatiou, A.; Chegkazi, M.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
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2013Sourcing the affinity of flavonoids for the glycogen phosphorylase inhibitor site via crystallography, kinetics and QM/MM-PBSA binding studies: Comparison of chrysin and flavopiridolTsitsanou K.E.; Hayes J.M.; Keramioti M.; Mamais M.; Oikonomakos N.G.; Kato A.; Leonidas D.D.; Zographos S.E.
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2014Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: Synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methodsCzifrák K.; Páhi A.; Deák S.; Kiss-Szikszai A.; Kövér K.E.; Docsa T.; Gergely P.; Alexacou K.-M.; Papakonstantinou M.; Leonidas D.D.; Zographos S.E.; Chrysina E.D.; Somsák L.
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2014Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-β-d-glucopyranosylaminesParmenopoulou V.; Kantsadi A.L.; Tsirkone V.G.; Chatzileontiadou D.S.M.; Manta S.; Zographos S.E.; Molfeta C.; Archontis G.; Agius L.; Hayes J.M.; Leonidas D.D.; Komiotis D.
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2019Anomeric spironucleosides of β-D-glucopyranosyl uracil as potential inhibitors of glycogen phosphorylaseStathi A.; Mamais M.; Chrysina E.D.; Gimisis T.
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2020Synthesis, kinetic and conformational studies of 2-substituted-5-(β-d-glucopyranosyl)-pyrimidin-4-ones as potential inhibitors of glycogen phosphorylaseMavreas, Konstantinos F; Neofytos, Dionysios D; Chrysina, Evangelia D. ; Venturini, Alessandro; Gimisis, Thanasis
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2021Glycogen phosphorylase revisited: Extending the resolution of the R- and T-state structures of the free enzyme and in complex with allosteric activatorsLeonidas, Demetres D; Zographos, S. E. ; Tsitsanou, K. E. ; Skamnaki, Vassiliki T; Stravodimos, George; Kyriakis, Efthimios
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2022Formation and physicochemical properties of glycogen phosphorylase in complex with a cationic polyelectrolyteNeofytos, Dionysios D; Papagiannopoulos, Aristeidis ; Chrysina, Evangelia D.; Pispas, Stergios
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