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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
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2008New Inhibitors of Glycogen Phosphorylase as Potential Antidiabetic AgentsSomsak, L.; Czifrak, K.; Toth, M.; Bokor, E.; Chrysina, Evangelia D.; Alexacou, K. -M.; Hayes, J. M.; Tiraidis, C.; Lazoura, E.; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.
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2008Naturally occurring pentacyclic triterpenes as inhibitors of glycogen phosphorylase: Synthesis, structure-activity relationships, and X-ray crystallographic studiesWen, Xiaoan; Sun, Hongbin; Liu, Jun; Cheng, Keguang; Zhang, Pu; Zhang, Liying; Hao, Jia; Zhang, Luyong; Ni, Peizhou; Zographos, Spyros E.; Leonidas, Demetres D.; Alexacou, Kyra-Melinda; Gimisis, Thanasis; Hayes, Joseph M.; Oikonomakos, Nikos G.
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2008Pentacyclic triterpenes, inhibitors of glycogen phosphorylase, as potential drugs for type 2 diabetes: X-ray crystallographic studiesZographos, Spyros E.; Leonidas, Demetres D.; Alexacou, K. M.; Gimisis, T.; Hayes, J. M.; Oikonomakos, Nikos G.; Wen, X.; Sun, H.; Liu, J.; Cheng, K.; Zhang, P.; Zhang, L.; Hao, J.; Zhang, L.; Ni, P.
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2009Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitorsBenltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Chrysina, Evangelia D.; Zographos, Spyros E.; Leonidas, Demetres D.; Archontis, Georgios; Oikonomakos, Nikos G.
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2009Morpholino, Piperidino, and Pyrrolidino Derivatives of Pyrimidine Nucleosides as Inhibitors of Ribonuclease A: Synthesis, Biochemical, and Crystallographic EvaluationSamanta, Anirban; Leonidas, Demetres D.; Dasgupta, Swagata; Pathak, Tanmaya; Zographos, Spyros E.; Oikonomakos, Nikos G.
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2008New synthetic seven-membered 1-azasugars displaying potent inhibition towards glycosidases and glucosylceramide transferaseLi, Hongqing; Liu, Tao; Zhang, Yongmin; Favre, Sylvain; Bello, Claudia; Vogel, Pierre; Butters, Terry D.; Oikonomakos, Nikos G.; Marrot, Jerome; Bleriot, Yves
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2006Indirubin and indigo analogues as potential inhibitors of glycogenolysis: structural basis of glycogen phosphorylase inhibitionOikonomakos, Nikos G.; Kosmopoulou, Magda N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Tiraidis, Costas; Bischler, Nicolas; Tsitsanou, Katerina E.; Zographos, Spyros E.; Kostas, Ioannis D.; Eisenbrand, Gerhard
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