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ΤύποςΗμερομηνίαΤίτλοςΔημιουργόςΠλήρες κείμενο
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2006Indirubin and indigo analogues as potential inhibitors of glycogenolysis: structural basis of glycogen phosphorylase inhibitionOikonomakos, Nikos G.; Kosmopoulou, Magda N.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Tiraidis, Costas; Bischler, Nicolas; Tsitsanou, Katerina E.; Zographos, Spyros E.; Kostas, Ioannis D.; Eisenbrand, Gerhard
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2008Advances in glycogen phosphorylase inhibitor designOikonomakos, Nikos G.; Somsak, Laszlo
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2008Crystallographic and computational studies on 4-phenyl-N-(beta-D-glucopyranosyl)-1H-1,2, 3-triazole-1-acetamide, an inhibitor of glycogen phosphorylase: Comparison with alpha-D-glucose, N-acetyl-beta-D-glucopyranosylamine and N-benzoyl-N '-beta-D-glucopyranosyl urea bindingAlexacou, Kyra-Melinda; Hayes, Joseph M.; Tiraidis, Costas; Zographos, Spyros E.; Leonidas, Demetres D.; Chrysina, Evangelia D.; Archontis, Georgios; Oikonomakos, Nikos G.; Paul, Jashuva V.; Varghese, Babu; Loganathan, Duraikkannu
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2009Glucose-based spiro-isoxazolines: A new family of potent glycogen phosphorylase inhibitorsBenltifa, Mahmoud; Hayes, Joseph M.; Vidal, Sebastien; Gueyrard, David; Goekjian, Peter G.; Praly, Jean-Pierre; Kizilis, Gregory; Tiraidis, Costas; Alexacou, Kyra-Melinda; Chrysina, Evangelia D.; Zographos, Spyros E.; Leonidas, Demetres D.; Archontis, Georgios; Oikonomakos, Nikos G.
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20101-(3-Deoxy-3-fluoro-beta-D-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studiesTsirkone, Vicky G.; Tsoukala, Evangelia; Lamprakis, Christos; Manta, Stella; Hayes, Joseph M.; Skamnaki, Vicky T.; Drakou, Christina; Zographos, Spyros E.; Komiotis, Dimitri; Leonidas, Demetres D.
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2010The Prototype of Glycogen PhosphorylaseChrysina, Evangelia D.
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2010The binding of beta-D-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitorsAlexacou, Kyra-Melinda; Tenchiu (Deleanu), Alia-Cristina; Chrysina, Evangelia D.; Charavgi, Maria-Despoina; Kostas, Ioannis D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2011Halogen-substituted (C-beta-D-glucopyranosyl)-hydroquinone regioisomers: Synthesis, enzymatic evaluation and their binding to glycogen phosphorylaseAlexacou, Kyra-Melinda; Zhang, Yun Zhi; Praly, Jean-Pierre; Zographos, Spyros E.; Chrysina, Evangelia D.; Oikonomakos, Nikos G.; Leonidas, Demetres D.
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2012N-(4-Substituted-benzoyl)-N '-(beta-D-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methodsVeronika Nagy; Nora Felfoeldi; Balint Konya; Praly, Jean-Pierre; Tibor Docsa; Pal Gergely; Chrysina, Evangelia D.; Tiraidis, Costas; Kosmopoulou, Magda N.; Alexacou, Kyra-Melinda; Konstantakaki, Maria; Leonidas, Demetres D.; Zographos, Spyros E.; Oikonomakos, Nikos G.; Kozmon, Stanislav; Tvaroska, Igor; Laszlo Somsak
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20123 '-Axial CH2OH Substitution on Glucopyranose does not Increase Glycogen Phosphorylase Inhibitory Potency. QM/MM-PBSA Calculations Suggest WhyManta, Stella; Xipnitou, Andromachi; Kiritsis, Christos; Kantsadi, Anastassia L.; Hayes, Joseph M.; Skamnaki, Vicky T.; Lamprakis, Christos; Kontou, Maria; Zoumpoulakis, Panagiotis; Zographos, Spyros E.; Leonidas, Demetres D.; Komiotis, Dimitri
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2014Structure based inhibitor design targeting glycogen phosphorylase b. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-β-d-glucopyranosylaminesParmenopoulou V.; Kantsadi A.L.; Tsirkone V.G.; Chatzileontiadou D.S.M.; Manta S.; Zographos S.E.; Molfeta C.; Archontis G.; Agius L.; Hayes J.M.; Leonidas D.D.; Komiotis D.
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2015Molecular cloning, carbohydrate specificity and the crystal structure of two Sclerotium rolfsii lectin variantsPeppa V.I.; Venkat H.; Kantsadi A.L.; Inamdar S.R.; Bhat G.G.; Eligar S.; Shivanand A.; Chachadi V.B.; Satisha G.J.; Swamy B.M.; Skamnaki V.T.; Zographos S.E.; Leonidas D.D.
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2017A New Potent Inhibitor of Glycogen Phosphorylase Reveals the Basicity of the Catalytic SiteMamais M.; Degli Esposti A.; Kouloumoundra V.; Gustavsson T.; Monti F.; Venturini A.; Chrysina E.D.; Markovitsi D.; Gimisis T.
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2018Structural features and catalytic reactivity of [Pd{(Ph2P)2N(CH2)3Si(OCH3)3-κP,P′}I2] and related complexes in hydroalkoxycarbonylation and Suzuki–Miyaura C−C cross-coupling reactionsStamatopoulos I.K.; Kapsi M.; Roulia M.; Vougioukalakis G.C.; Raptopoulou C.P.; Psycharis V.; Kostas I.D.; Kollár L.; Kyritsis P.
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2020The crystal structure of a Fusarium oxysporum feruloyl esterase that belongs to the tannase familyDimarogona, Maria; Topakas, Evangelos; Christakopoulos, Paul; Evangelia D. Chrysina
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